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Cat.No. Product Name / Introduction Added
CS-3535 PRT062607 December 2014
PRT062607(P505-15; PRT-2607; BIIB-057) is a highly specific and potent inhibitor of Syk with IC50 of 1-2 nM; >80-fold selective for Syk than Fgr, Lyn, FAK, Pyk2 and Zap70.
 
CS-3530 Stauprimide December 2014
Stauprimide is a small molecule that increases the efficiency of the directed differentiation of mouse and human ESCs; interacts with NME2 and inhibits its nuclear localization.
 
CS-3544 BQ-788 December 2014
BQ-788 is a potent and selective endothelin receptor subtype B (ETB) antagonist with IC50 of 1.
 
CS-3538 SB225002 December 2014
SB225002 is a potent and selective non-peptide inhibitor of CXCR2 with IC50 of 22 nM; >150-fold selectivity over CXCR1 and four other 7-TMRs.
 
CS-3545 Apoptosis-Activator-2 December 2014
Apoptosis Activator 2 is a potent apoptosis activator; increases procaspase-9 processing and subsequent caspase-3 activation.
 
CS-3543 Promethazine-hydrochloride December 2014
Promethazine Hcl(NSC-231688) is the first-generation antihistamine; strong antagonist of the H1 receptor and moderate mACh receptor antagonist, moderate affinity for 5-HT2A, 5-HT2C, D2 and α1-adrenergic receptors.
 
CS-3542 NSC319726 December 2014
NSC319726 is a mutant p53R175 reactivator; inhibits growth of fibroblasts expressing the p53R175 mutation (IC50 = 8 nM); shows no inhibition for p53 wild-type cells.
 
CS-3541 Lucigenin December 2014
Lucigenin(L-6868; NSC-151912) is a chemiluminescent probe used to indicate the presence of endogenously generated superoxide anion radicals in cells.
 
CS-3540 Fluorescein-Diacetate December 2014
Fluorescein diacetate(Di-O-acetylfluorescein) is a cell-permeant esterase substrate that can serve as a viability probe that measures both enzymatic activity, which is require to activate its fluorescence, and cell-membrane integrity, which is required for intracellular retention of their fluorescent product.
 
CS-3539 1627503-67-6 December 2014
LDN-214117 is a potent and selective ALK2 inhibitor with IC50 of 22 nM; > 100 fold selectivity for ALK5; also inhibits BMP6(IC50=100 nM).
 
CS-3537 CWHM-12 December 2014
CWHM-12 a novel small molecule inhibitor of αV integrins with IC50s of 1.
 
CS-3536 TZ9 December 2014
TZ9 is a novel inhibitor of Rad6 ubiquitin conjugating enzyme(E2 enzyme); inhibits MDA-MB-231 cell proliferation with IC50 of ~6 uM.
 
CS-3534 K-Ras-G12C-IN-3 December 2014
K-Ras G12C-IN-3 is a novel and irreversible inhibitor of mutant K-ras G12C.
 
CS-3533 K-Ras-G12C-IN-2 December 2014
K-Ras G12C-IN-2 is a novel and irreversible inhibitor of mutant K-ras G12C.
 
CS-3532 K-Ras-G12C-IN-1 December 2014
K-Ras G12C-IN-1 is a novel and irreversible inhibitor of mutant K-ras G12C.
 
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CS-0757 SB-705498
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CS-0765 CYT387 sulfate salt
CYT387 sulfate(momelotinib) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, ~10-fold selectivity versus JAK3.
CS-0645 Rimonabant
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CS-0494 XAV-939
XAV939 is a small molecule and selective Wnt pathway β-catenin-mediated transcription inhibitor and axin stabilizing agent with IC50 of 11 and 4 nM for the inhibition of TNKS1 and TNKS2, respectively.
CS-0264 DAPT
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CS-0361 Boceprevir
Boceprevir(EBP-520, SCH503034) is an HCV protease inhibitor (Ki=14 nM) for the treatment of hepatitis C virus infection.
CS-0592 YM-201636
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CS-0613 Tideglusib
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CS-0625 Avosentan
Avosentan(Ro 67-0565; SPP-301) is a potent, selective endothelin receptor(ETA receptor) antagonist.
CS-0609 SCH 527123
SCH-527123 is a potent antagonist of both CXCR1 and CXCR2 with IC50 of 42 nM and 3 nM, respectively.
CS-0612 T 705
T 705 (Favipiravir) is an experimental anti-viral drug with activity against many RNA viruses; RNA-directed RNA polymerase NS5B inhibitor.
CS-0614 Suvorexant
Suvorexant (MK-4305) is a potent dual OX receptor antagonist with Ki of 0.
CS-0627 MEK162
MEK162(ARRY-438162; ARRY-162) is a potent inhibitor of MEK1/2 with IC50 of 12 nM.
CS-0608 BMS-754807
BMS-754807 is a potent and reversible inhibitor of IGF-1R/InsR with IC50 of 1.

 
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