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Cat.No. Product Name / Introduction Added
CS-6033 Sophoflavescenol December 2016
Sophoflavescenol is a prenylated flavonol, which shows great inhibitory activity with IC50 of 13 nM against Phosphodiesterase 5 (PDE5), and also inhibits RLAR, HRAR, AGE, BACE1, AChE and BChE with IC50s of 0.
 
CS-6052 Phorbol December 2016
Phorbol is a highly toxic diterpene, and it's esters have important biological properties.
 
CS-6051 Epoxymicheliolide December 2016
Epoxymicheliolide is a micheliolide derivative.
 
CS-6050 Protodioscin December 2016
Protodioscin, a major steroidal saponin in dioscoreae rhizome, has been shown to exhibit multiple biological actions, such as anti-hyperlipidemia, anti-cancer, sexual effects and cardiovascular properties.
 
CS-6049 Hederacoside-D December 2016
Hederacoside D is one of the bioactive saponins from Hedera helix, and plays pivotal roles in the overall biological activity.
 
CS-4274 Tanshinone-I December 2016
Tanshinone I is an inhibitor of type IIA human recombinant sPLA2(IC50=11 μM) and rabbit recombinant cPLA2(IC50=82 μM).
 
CS-6053 Phorbol-12-myristate-13-acetate December 2016
Phorbol 12-myristate 13-acetate (PMA) is a PKC-activating phorbol ester, increases the intracellular Ca2+ concentration ([Ca2+]i) in a dose-dependent manner, with an EC50 of 11.
 
CS-6046 Basmisanil December 2016
Basmisanil is a highly selective GABAAα5 negative allosteric modulator.
 
CS-6048 Bromocriptine-mesylate December 2016
Bromocriptine mesylate is a potent dopamine D2/D3 receptor agonist, which binds D2 dopamine receptor with pKi of 8.
 
CS-6041 Beclabuvir December 2016
Beclabuvir is an allosteric inhibitor that binds to thumb site 1 of the hepatitis C virus (HCV) NS5B RNA-dependent RNA polymerase, and inhibits recombinant NS5B proteins from HCV genotypes 1, 3, 4, and 5 with IC50 of < 28 nM.
 
CS-6047 YM-58483 December 2016
YM-58483 is the first selective and potent inhibitor of CRAC channels and subsequent Ca2+ signals.
 
CS-6045 BGP-15 December 2016
BGP-15 is a PARP inhibitor, that can protect against heart failure and atrial fibrillation in mice.
 
CS-6043 Ribitol December 2016
Ribitol is a crystalline pentose alcohol formed by the reduction of ribose.
 
CS-6044 BFH772 December 2016
BFH772 is a potent oral VEGFR2 inhibitor, which is highly effective at targeting VEGFR2 kinase with an IC50 value of 3 nM.
 
CS-6040 SKF89976A-hydrochloride December 2016
SKF89976A hydrochloride is a selective GABA transporter (GAT-1) inhibitor with IC50s of 0.
 
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CS-0645 Rimonabant
Rimonabant(SR141716) is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.
CS-2222 Meprednisone
Meprednisone is a glucocorticoid and a methylated derivative of prednisone.
CS-0264 DAPT
DAPT(GSI-IX) is an inhibitor of γ-secretase; DAPT causes a reduction in Aβ40 and Aβ42 levels in human primary neuronal cultures (IC50 values are 115 and 200 nM for total Aβ and Aβ42 respectively) and in brain extract, cerebrospinal fluid and plasma in vivo.
CS-0613 Tideglusib
Tideglusib(NP-031112) is an irreversible, non ATP-competitive GSK-3β inhibitor with IC50 of 60 nM.
CS-0757 SB-705498
SB-705498 is a potent, selective and orally bioavailable transient receptor potential vanilloid 1 (TRPV1) receptor antagonist with a pIC50 of 7.
CS-0766 Aripiprazole
Aripiprazole(Abilify) is a human 5-HT1A receptor partial agonist with a Ki of 4.
CS-1971 Haloperidol
Haloperidol blocks dopamine receptors in in the treatment of schizophrenia, acute psychosis, and delirium.
CS-0609 SCH 527123
SCH-527123 is a potent antagonist of both CXCR1 and CXCR2 with IC50 of 42 nM and 3 nM, respectively.
CS-0361 Boceprevir
Boceprevir(EBP-520, SCH503034) is an HCV protease inhibitor (Ki=14 nM) for the treatment of hepatitis C virus infection.
CS-0625 Avosentan
Avosentan(Ro 67-0565; SPP-301) is a potent, selective endothelin receptor(ETA receptor) antagonist.
CS-0494 XAV-939
XAV939 is a small molecule and selective Wnt pathway β-catenin-mediated transcription inhibitor and axin stabilizing agent with IC50 of 11 and 4 nM for the inhibition of TNKS1 and TNKS2, respectively.
CS-0592 YM-201636
YM201636 is a selective PIKfyve inhibitor with IC50 of 33 nM, less potent to p110α.
CS-0608 BMS-754807
BMS-754807 is a potent and reversible inhibitor of IGF-1R/InsR with IC50 of 1.
CS-0627 MEK162
MEK162(ARRY-438162; ARRY-162) is a potent inhibitor of MEK1/2 with IC50 of 12 nM.
CS-0765 CYT387 (sulfate salt)
CYT387 sulfate(momelotinib) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, ~10-fold selectivity versus JAK3.
CS-1955 CC-401
CC-401 is a second generation ATP-competitive anthrapyrazolone c-Jun N terminal kinase (JNK) inhibitor with potential antineoplastic activity.
CS-1956 XL413
XL413 is a potent and selective Cdc7 inhibitor with an IC50 of 3.
CS-B0575 1H-Pyrrolo[2,3-b]pyridin-4-amine, 1-methyl-
CS-B0576 1H-Pyrrolo[2,3-b]pyridine-1-carboxylic acid, 4-amino-, 1,1-dimethylethyl ester
CS-B0577 1H-Pyrrolo[2,3-b]pyridin-4-amine, 1-(phenylmethyl)-

 
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