ADL-5859 M.Wt: 428.95
ADL-5859 Formula: C24H29ClN2O3
ADL-5859 Solubility: DMSO ≥84mg/mL Water ≥10mg/mL Ethanol ≥0.8mg/mL
ADL-5859 Purity: >98%
Please store the product under the recommended conditions in the Certificate of Analysis.
ADL5859 is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel.
IC50 value: 0.8 nM(Ki)
Target: δ-opioid receptor
ADL-5859 (ADL5859) is an δ-opioid receptor agonist (Ki=0.84 nM, EC50=20 nM). ADL-5859 (ADL5859) is an agonist agent that selectively stimulates the δ-opioid receptor with potential application in a wide range of inflammatory, neuropathic and acute pain conditions. In addition, Delta agonists are thought to modulate other biological processes that may manifest themselves in disease states or conditions such as overactive bladder and depression.ADL-5859 (ADL5859) is useful for inflammatory, neuropathic and acute pain conditions.