Lot numbers can be found on the outside label of a product:
Please log in for operation!
*For research and further manufacturing use only, not for direct human use.
Structure of 877399-31-0
| Size |
|
Price | Quantity | |||
|---|---|---|---|---|---|---|
|
* Please select Quantity before adding items. |
||||||
tert-Butyl 3-{[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]methyl}azetidine-1-carboxylate features a pyrazole-borane moiety integrated with a sterically shielded azetidine scaffold, delivering enhanced stability and reactivity in Suzuki-Miyaura coupling processes. The tetramethylboronate group enables efficient cross-coupling under mild conditions, while the tert-butyl ester ensures compatibility with standard deprotection workflows. This compound serves as a modular building block for complex heterocyclic architectures in medicinal chemistry and materials science.
tert-Butyl 3-{[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]methyl}azetidine-1-carboxylate serves as a versatile boron-containing building block for Suzuki-Miyaura cross-coupling reactions. The azetidine core provides a strained, bioactive scaffold, while the pyrazole moiety offers hydrogen-bonding capacity and metabolic stability. The tert-butyl carbamate group enables mild deprotection under acidic conditions, facilitating downstream functionalization. This compound exhibits excellent bench stability, tolerates diverse reaction conditions, and is readily purified by standard chromatography, making it ideal for iterative medicinal chemistry campaigns and API intermediate synthesis.
|
GHS Pictogram :
|
GHS No : GHS07
|
|
Signal Word : Warning
|
UN#: N/A
|
|
Class : N/A
|
Packing Group : N/A
|
|
Hazard Statements : H302-H315-H319-H335
|
|
|
Precautionary Statements : P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P403+P233-P405-P501
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
Upload Pictures
|
|
Lot numbers can be found on the outside label of a product: